SCHEMBL28630576

SCHEMBL28630576

CCOC(=O)C=CC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
MAOB P27338 4/20 0.56
CES2 O00748 1/20 0.50
POLB P06746 1/20 0.49
MAPT P10636 5/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADORA1 P30542 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24951715 1.00 ALDH1A1 (0.59) ALDH1A1MAOBCES2POLBMAPT
Ethyl Fumarate SCHEMBL8787704 0.84 HCAR2 (0.48) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL10399108 0.83 CES2 (0.47) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL10399189 0.83 CES2 (0.47) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL10399109 0.83 CES2 (0.47) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL29098730 0.83 CYP1A1 (0.58) MAOBMAPTNPSR1
SCHEMBL3269421 0.82 NPSR1 (0.52) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL7361886 0.82 ALDH1A1 (0.60) ALDH1A1MAOBCES2POLBMAPT
SCHEMBL29098722 0.81 MAPT (0.54) ALDH1A1MAPTLMNA
SCHEMBL30786693 0.81 CES2 (0.61) ALDH1A1CES2POLBMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113444081-B Thiadiazole carboxamide compounds and application thereof 浙江大学 2022-07-05 CN disclosed
CN-113444081-A Thiadiazole amide compound and application thereof 浙江大学 2021-09-28 CN disclosed