SCHEMBL7362256

SCHEMBL7362256

CC(C)C[C](Cc1ccccc1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
AKR1B1 P15121 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
TRPA1 O75762 1/20 0.39
PSMB8 P28062 1/20 0.39
PSMB5 P28074 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A2 P23975 2/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAOA P21397 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CYP2A6 P11509 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369705 0.87 TSHR (0.50) TSHRCES2CES1AKR1B1KMT2A
SCHEMBL7394095 0.77 TSHR (0.46) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL106992 0.75 TSHR (0.53) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL11908722 0.74 TSHR (0.47) TSHRCES2CES1AKR1B1ALDH1A1
Phenylacetic Acid SCHEMBL28235727 0.73 AKR1B1 (0.68) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL448700 0.73 CES2 (0.68) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL3245857 0.73 TSHR (0.50) TSHRCES2CES1AKR1B1KMT2A
SCHEMBL9354964 0.72 TSHR (0.50) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL9355881 0.72 TSHR (0.50) TSHRCES2CES1AKR1B1ALDH1A1
SCHEMBL7361543 0.72 MAOA (0.46) TSHRKMT2ASMN1; SMN2SLC6A2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722321-A4 SULFOXIMINE AND SULFODIIMINE MATRIX METALLOPROTEINASE INHIBITORS UNIV FLORIDA STATE (US) 1998-04-15 EP disclosed
EP-0722321-A1 SULFOXIMINE AND SULFODIIMINE MATRIX METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1996-07-24 EP disclosed
WO-1995009620-A1 SULFOXIMINE AND SULFODIIMINE MATRIX METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1995-04-13 WO disclosed