SCHEMBL7362905

SCHEMBL7362905

CCOC(=O)CNCCCC(c1ccc(N)cc1)c1cccc(C(=N)N)c1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
F10 P00742 17/20 0.53
F2 P00734 16/20 0.51
PRSS1 P07477 9/20 0.51
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6006300 0.80 LTA4H (0.56) LTA4H
SCHEMBL6005586 0.72 LTA4H (0.53) LTA4H
SCHEMBL7360130 0.72 F10 (0.58) F10F2PRSS1
SCHEMBL7365375 0.71 F10 (0.56) F10F2PRSS1
SCHEMBL8346836 0.70 F10 (0.49) F10F2PRSS1LTA4H
SCHEMBL7455464 0.68 F10 (1.00) F10F2PRSS1
Trifluoroacetic Acid SCHEMBL8343413 0.67 F2 (0.48) F10F2PRSS1LTA4H
SCHEMBL1624623 0.67 F10 (0.54) F10F2PRSS1
SCHEMBL7460126 0.67 F10 (0.63) F10F2PRSS1
SCHEMBL5691956 0.66 ALDH1A1 (0.59) F10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed