SCHEMBL7363403

SCHEMBL7363403

N#Cc1cccc(N)c1CCCCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
KCNH2 Q12809 5/20 0.43
KCNJ1 P48048 4/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
TSHR P16473 1/20 0.41
VCAM1 P19320 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
KMT2A Q03164 1/20 0.39
RAB9A P51151 1/20 0.39
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7363839 0.81 CYP1A2 (0.33) CASP3SENP8SENP7SENP6
SCHEMBL18913824 0.73 TSHR (0.69) KCNH2KCNJ1LOXL2TSHRSIGMAR1
Methylamine SCHEMBL27524577 0.73 SIGMAR1 (0.61) KCNH2KCNJ1LOXL2TSHRSIGMAR1
SCHEMBL6089703 0.71 CYP3A4 (0.42) KCNH2TSHRMAPTALDH1A1
SCHEMBL9640859 0.71 KCNH2 (0.68) KCNH2KCNJ1LOXL2TSHRVCAM1
Dinitrophenylene SCHEMBL27864502 0.70 TSHR (0.57) CASP3SENP8SENP7SENP6TSHR
SCHEMBL30758863 0.70 TSHR (0.69) KCNH2KCNJ1LOXL2TSHRSIGMAR1
SCHEMBL9055361 0.70 TSHR (0.55) KCNH2KCNJ1LOXL2TSHRSIGMAR1
SCHEMBL6481704 0.69 ALDH1A1 (0.69) KCNH2KCNJ1LOXL2TSHRSIGMAR1
SCHEMBL1163856 0.69 SIGMAR1 (0.65) KCNH2KCNJ1LOXL2TSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed