SCHEMBL7363690

SCHEMBL7363690

CCCCCc1ccnc(N2CCNCC2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.54
ADRB1 P08588 1/20 0.49
HRH4 Q9H3N8 3/20 0.48
NMT1 P30419 6/20 0.46
PLD1 Q13393 1/20 0.45
MAOB P27338 1/20 0.43
HTR6 P50406 1/20 0.43
DYRK1A Q13627 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRL1 P41146 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11546296 0.90 AOC3 (0.57) AOC3ADRB1HRH4NMT1PLD1
SCHEMBL11919149 0.84 ADRB1 (0.55) AOC3ADRB1HRH4NMT1PLD1
SCHEMBL21376960 0.83 PIK3CA (0.50) OPRM1OPRL1
Hydrochloric Acid SCHEMBL31061226 0.82 ADRB1 (0.54) AOC3ADRB1HRH4NMT1PLD1
SCHEMBL13361855 0.78 ADRB1 (0.59) AOC3ADRB1HRH4NMT1PLD1
SCHEMBL2328273 0.78 AOC3 (0.56) AOC3ADRB1HRH4NMT1PLD1
SCHEMBL3640716 0.78 HRH3 (0.52) ADRB1HRH4PLD1HTR6HRH3
SCHEMBL4563936 0.78 HTR2C (0.37) AOC3HRH4HTR2AHTR2C
SCHEMBL15621623 0.76 HRH4 (0.49) AOC3HRH4OPRM1OPRL1
SCHEMBL23630504 0.76 AOC3 (0.60) AOC3ADRB1HRH4NMT1PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385237-B1 2-(1-piperazinyl)-4-phenylcycloalkanopyridine derivatives, processes for the production thereof, and pharmaceutical composition containing the same DAINIPPON PHARMACEUTICAL CO (JP) 1994-06-29 EP disclosed
US-5021421-A Psychotropic agents DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1991-06-04 US disclosed
EP-0385237-A2 2-(1-piperazinyl)-4-phenylcycloalkanopyridine derivatives, processes for the production thereof, and pharmaceutical composition containing the same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1990-09-05 EP disclosed