SCHEMBL7364062

SCHEMBL7364062

CC1(C)OCC(Cc2ccc(OCC(F)(F)F)cc2)N1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PPARG P37231 4/20 0.36
PPARA Q07869 3/20 0.36
LMNA P02545 2/20 0.36
PMP22 Q01453 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXRA P19793 1/20 0.36
HNF4A P41235 1/20 0.36
CYP1A2 P05177 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2B P41595 1/20 0.35
KCNH2 Q12809 1/20 0.35
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35
LIPE Q05469 2/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6540867 0.84 PPARA (0.39) SMN1; SMN2PPARGPPARAALDH1A1CYP3A4
SCHEMBL6540875 0.84 PPARA (0.39) SMN1; SMN2PPARGPPARAALDH1A1CYP3A4
SCHEMBL7364066 0.81 PPARA (0.38) SMN1; SMN2NPC1RAB9APPARGPPARA
SCHEMBL6541438 0.80 CAPN1 (0.38) SMN1; SMN2PPARGALDH1A1CYP3A4HPGD
SCHEMBL6541442 0.80 CAPN1 (0.38) SMN1; SMN2PPARGALDH1A1CYP3A4HPGD
SCHEMBL6539634 0.78 MAPT (0.38) SMN1; SMN2PPARGALDH1A1CYP3A4HPGD
SCHEMBL6539645 0.78 MAPT (0.38) SMN1; SMN2PPARGALDH1A1CYP3A4HPGD
SCHEMBL6539667 0.78 PTGIR (0.41) SMN1; SMN2NPC1RAB9ALMNANPSR1
SCHEMBL6540931 0.78 PKM (0.44) SMN1; SMN2LMNANPSR1CYP2C19MMP13
SCHEMBL6539664 0.78 PTGIR (0.41) SMN1; SMN2NPC1RAB9ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194404-A1 INHIBITORS OF ASPARTYL PROTEASE Vertex Pharmaceuticals Incorporated (US) 2002-04-10 EP disclosed
WO-2000076961-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-12-21 WO disclosed