SCHEMBL7364066

SCHEMBL7364066

CN1C(Cc2ccc(OCC(F)(F)F)cc2)COC1(C)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 9/20 0.38
PPARG P37231 9/20 0.38
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
CYP1A2 P05177 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2B P41595 1/20 0.35
KCNH2 Q12809 1/20 0.35
LIPE Q05469 2/20 0.34
FFAR1 O14842 1/20 0.34
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364062 0.81 SMN1; SMN2 (0.37) PPARAPPARGCARM1PRMT6CYP1A2
Bicarbonate SCHEMBL27771212 0.66 SMN1; SMN2 (0.51) CYP1A2CYP2C19NPC1RAB9ASMN1; SMN2
SCHEMBL6540867 0.66 PPARA (0.39) PPARAPPARGSMN1; SMN2
SCHEMBL6540875 0.66 PPARA (0.39) PPARAPPARGSMN1; SMN2
SCHEMBL964774 0.64 RXRA (0.50) PPARAPPARGKCNH2NPC1RAB9A
SCHEMBL2714295 0.62 MAOB (0.62) MAOBNPC1RAB9ASMN1; SMN2
SCHEMBL28901155 0.62 LIPE (0.43) PPARACARM1PRMT6LIPENPC1
SCHEMBL31258914 0.62 PTPN1 (0.65) PPARAPPARGCYP1A2HTR2AKCNH2
SCHEMBL13957613 0.62 PTPN1 (0.65) PPARAPPARGCYP1A2HTR2AKCNH2
SCHEMBL23052638 0.61 PPARA (0.47) PPARAPPARGCYP1A2KCNH2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194404-A1 INHIBITORS OF ASPARTYL PROTEASE Vertex Pharmaceuticals Incorporated (US) 2002-04-10 EP disclosed
WO-2000076961-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-12-21 WO disclosed