SCHEMBL7364095

SCHEMBL7364095

Nc1n[nH]cc1-c1ccoc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.42
STK4 Q13043 1/20 0.40
STK3 Q13188 1/20 0.40
FYN P06241 5/20 0.38
CDK8 P49336 1/20 0.37
CSNK2A1 P68400 1/20 0.36
ADORA2A P29274 1/20 0.36
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2D6 P10635 3/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2E1 P05181 2/20 0.35
CYP2A6 P11509 2/20 0.35
CYP2B6 P20813 2/20 0.35
CYP2C8 P10632 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065086 0.74 IMPDH2 (0.44) IMPDH2STK4STK3FYNCDK8
SCHEMBL544598 0.71 MAP4K4 (0.48) CYP1A2ALDH1A1HSD17B10CLK4
SCHEMBL3724188 0.71 KDR (0.46) CYP3A4CHEK1ALDH1A1HSD17B10
SCHEMBL18613440 0.70 FYN (0.53) IMPDH2FYNCDK8CYP1A2CYP3A4
SCHEMBL1925085 0.69 IMPDH2 (0.43) IMPDH2CDK8CYP1A2CYP3A4CYP2D6
SCHEMBL21223675 0.69 CYP1A2 (0.42) IMPDH2FYNCSNK2A1ADORA2ACDK2
SCHEMBL17555670 0.69 FYN (0.41) FYNCSNK2A1ADORA2ACCNT1CCNA2
SCHEMBL17619924 0.68 MAPK14 (0.49) STK4STK3ADORA2AALDH1A1CLK4
SCHEMBL9735461 0.68 IKBKB (0.46) CYP1A2ALDH1A1
SCHEMBL6487188 0.66 GSK3B (0.57) CSNK2A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed