SCHEMBL9735461

SCHEMBL9735461

Nc1n[nH]cc1-c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.46
MAP3K14 Q99558 1/20 0.46
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
ALPL P05186 1/20 0.44
TDO2 P48775 1/20 0.44
MAP4K4 O95819 8/20 0.43
CYP1A2 P05177 1/20 0.42
KCNH2 Q12809 1/20 0.42
MINK1 Q8N4C8 1/20 0.42
TNIK Q9UKE5 1/20 0.42
LTA4H P09960 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ABL1 P00519 1/20 0.40
SRC P12931 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724188 0.83 KDR (0.46) ALPLNPC1RAB9AABL1KDM4E
SCHEMBL13264574 0.81 AKT2 (0.60) IKBKBMAP3K14MAP4K4
SCHEMBL17619924 0.79 MAPK14 (0.49) MKNK1MKNK2TDO2MAP4K4RAB9A
SCHEMBL544598 0.78 MAP4K4 (0.48) MKNK1MKNK2TDO2MAP4K4CYP1A2
SCHEMBL24962591 0.78 IKBKB (0.41) IKBKBMAP3K14NPC1RAB9A
SCHEMBL7096615 0.78 KMT2A (0.38) CYP1A2NPC1RAB9AKDM4EHPGD
SCHEMBL1925085 0.77 IMPDH2 (0.43) CYP1A2NPC1RAB9AKDM4EALDH1A1
SCHEMBL1247672 0.75 KIF11 (0.48) MKNK1MKNK2MAP4K4NPC1RAB9A
SCHEMBL5872525 0.75 HSP90AA1 (0.45) ALPLRAB9AKDM4EALDH1A1HPGD
SCHEMBL22425324 0.73 ALDH1A1 (0.39) CYP1A2NPC1RAB9AABL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132424-A Anticholesterol, treatment of atherosclerosis THE UPJOHN COMPANY (US) 1992-07-21 US disclosed
EP-0425541-A1 PYRAZOLO-AZOLO-PYRIMIDINE-DIONES THE UPJOHN COMPANY (US) 1991-05-08 EP disclosed
WO-1990001031-A1 PYRAZOLO-PYRROLO-PYRIMIDINE-DIONES THE UPJOHN COMPANY (US) 1990-02-08 WO disclosed