SCHEMBL7364277

SCHEMBL7364277

Cc1cc(O)nc(NC2CCC(C)CC2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 10/20 0.40
ADRA2A P08913 3/20 0.40
HRH1 P35367 3/20 0.40
ADRA1A P35348 2/20 0.40
HTR2B P41595 2/20 0.40
DNM2 P50570 1/20 0.40
CNR1 P21554 1/20 0.39
KCNH2 Q12809 1/20 0.39
AURKB Q96GD4 1/20 0.39
KDM4E B2RXH2 2/20 0.39
GRM5 P41594 1/20 0.39
PTGS2 P35354 1/20 0.39
PI4KB Q9UBF8 1/20 0.38
LMNA P02545 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357755 0.81 MCHR1 (0.43) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL2369879 0.80 DNM2 (0.49) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL4908497 0.80 KDM4E (0.38) MCHR1KDM4E
SCHEMBL25920566 0.79 MCHR1 (0.42) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL25920567 0.77 CNR1 (0.45) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL1178837 0.71 MCHR1 (0.45) MCHR1ADRA2AHRH1ADRA1AHTR2B
SCHEMBL1334607 0.69 GRM5 (0.39) DNM2CNR1KCNH2AURKBKDM4E
SCHEMBL1334609 0.69 GRM5 (0.39) DNM2CNR1KCNH2AURKBKDM4E
SCHEMBL2276674 0.69 PLK4 (0.46) DNM2KDM4EPTGS2CYP1A2ATM
SCHEMBL10285741 0.69 MAPT (0.46) KDM4ELMNAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000027826-A1 NOVEL PYRIMIDINES, THE PRODUCTION THEREOF AND THEIR USE BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-05-18 WO disclosed