SCHEMBL7364494

SCHEMBL7364494

[CH2]c1cccc(CCCO)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 4/20 0.46
CYP4A11 Q02928 4/20 0.46
TBXA2R P21731 1/20 0.41
LTA4H P09960 1/20 0.41
EPHX2 P34913 1/20 0.41
TDP1 Q9NUW8 1/20 0.38
NOS1 P29475 1/20 0.38
IGF1R P08069 1/20 0.37
ALOX15 P16050 1/20 0.37
LPL P06858 2/20 0.37
LIPG Q9Y5X9 2/20 0.37
CA2 P00918 1/20 0.36
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10903519 0.94 CYP4F2 (0.50) CYP4F2CYP4A11TBXA2RTDP1NOS1
SCHEMBL10903699 0.92 CYP4F2 (0.49) CYP4F2CYP4A11IGF1RALOX15LPL
SCHEMBL577119 0.87 TDP1 (0.52) CYP4F2CYP4A11TDP1NOS1CA2
SCHEMBL241880 0.84 CYP4F2 (0.53) CYP4F2CYP4A11TBXA2RLTA4HEPHX2
SCHEMBL9501401 0.79 TAAR1 (0.35) NOS1IGF1RALOX15LPLLIPG
SCHEMBL9200094 0.79 TAAR1 (0.39) NOS1LPLLIPGDRD2DRD1
SCHEMBL613331 0.79 TAAR1 (0.48) CYP4F2CYP4A11TBXA2RLTA4HEPHX2
SCHEMBL5459240 0.79 LPL (0.49) TDP1LPLLIPGDRD2
SCHEMBL1244841 0.78 CYP4F2 (0.49) CYP4F2CYP4A11TBXA2RLTA4HEPHX2
SCHEMBL238401 0.78 CYP4F2 (0.58) CYP4F2CYP4A11TBXA2RTDP1NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
WO-1996029329-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-26 WO claimed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed
WO-1996029329-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-26 WO disclosed
US-4590291-A Thrombin inhibitory new dihydroxybenzene ether derivatives BAYER AKTIENGESELLSCHAFT (DE) 1986-05-20 US disclosed
EP-0068250-A1 Dioxybenzene ether derivatives, pharmaceutical compositions containing them, process for the preparation thereof and their use BAYER AG (DE) 1983-01-05 EP disclosed