SCHEMBL7364560

SCHEMBL7364560

COc1ccc(S(=O)(=O)N2Cc3cccc(Br)c3C2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.61
CYP2C19 P33261 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
GPBAR1 Q8TDU6 1/20 0.56
TSHR P16473 3/20 0.54
POLB P06746 2/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 2/20 0.52
LMNA P02545 2/20 0.52
USP2 O75604 1/20 0.52
GLA P06280 1/20 0.52
MAPK1 P28482 1/20 0.52
MCOLN3 Q8TDD5 2/20 0.50
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757285 0.79 PKM (0.51) CYP2C19SMN1; SMN2TSHRPOLBHTT
SCHEMBL28485965 0.77 CYP3A4 (0.49) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL28485032 0.77 CYP3A4 (0.49) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL3830421 0.77 GPBAR1 (0.90) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL4184681 0.77 GPBAR1 (0.90) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL28488424 0.77 CYP3A4 (0.48) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL6186477 0.77 HTR6 (0.58) CYP3A4CYP2C19SMN1; SMN2NPSR1TSHR
SCHEMBL6429647 0.76 CYP3A4 (1.00) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL28482926 0.75 CYP3A4 (0.49) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1
SCHEMBL28492863 0.75 CYP3A4 (0.49) CYP3A4CYP2C19SMN1; SMN2NPSR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996036611-A1 3,4-DISUBSTITUTED-PHENYLSULPHONAMIDES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed
US-5728712-A 3,4-disubstituted-phenylsulphonamides and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-03-17 US disclosed
WO-1996036611-A1 3,4-DISUBSTITUTED-PHENYLSULPHONAMIDES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO disclosed