SCHEMBL7364847

SCHEMBL7364847

O=Cc1cnn2c(-c3ccncc3)ccnc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.55
ALDH1A1 P00352 3/20 0.55
NPC1 O15118 2/20 0.55
MAPT P10636 2/20 0.55
RAB9A P51151 2/20 0.55
NFKB1 P19838 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
KDM4E B2RXH2 3/20 0.45
CLK4 Q9HAZ1 2/20 0.45
MAP2K1 Q02750 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MARK2 Q7KZI7 2/20 0.38
PDPK1 O15530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11482468 0.88 CLK4 (0.58) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL7361403 0.84 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL4702080 0.77 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL11350246 0.76 NPC1 (0.67) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL3172246 0.75 KDM4E (0.65) KDM4E
SCHEMBL29935834 0.74 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1NPC1RAB9AKDM4E
SCHEMBL14264668 0.74 MAPT (0.36) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL14264667 0.74 KDM4E (0.36) ALDH1A1NPC1RAB9AKDM4ECLK4
SCHEMBL9868803 0.74 MAP2K1 (0.80) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL11346886 0.73 KDM4E (0.78) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed