SCHEMBL7365569

SCHEMBL7365569

C=CC(=O)c1cccc(-c2cccnc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.67
P4HB P07237 1/20 0.53
MKNK1 Q9BUB5 7/20 0.51
MKNK2 Q9HBH9 7/20 0.51
MEN1 O00255 1/20 0.51
PSIP1 O75475 1/20 0.51
AXL P30530 1/20 0.51
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP2A6 P11509 1/20 0.47
ERN1 O75460 1/20 0.47
ABCB1 P08183 2/20 0.46
AKT1 P31749 1/20 0.46
USP2 O75604 1/20 0.46
CYP1A1 P04798 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP1B1 Q16678 2/20 0.45
CYP19A1 P11511 1/20 0.45
CYP11B1 P15538 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16111856 0.86 KMO (0.69) KMOP4HBMKNK1MKNK2MEN1
SCHEMBL27605046 0.82 KMO (0.77) KMOP4HBMKNK1MKNK2MEN1
SCHEMBL1583591 0.81 ALDH1A1 (0.59) MEN1CYP1A2CYP3A4ALDH1A1AKT1
SCHEMBL8431770 0.81 AKT1 (0.57) KMOMEN1CYP3A4ALDH1A1ERN1
SCHEMBL29569537 0.80 KMO (1.00) KMOMKNK1MKNK2MEN1PSIP1
SCHEMBL28297133 0.80 KMO (1.00) KMOMKNK1MKNK2MEN1PSIP1
SCHEMBL206541 0.80 KMO (1.00) KMOMKNK1MKNK2MEN1PSIP1
SCHEMBL30114603 0.80 KMO (0.65) KMOP4HBMKNK1MKNK2MEN1
SCHEMBL205967 0.79 KMO (0.73) KMOP4HBMKNK1MKNK2MEN1
SCHEMBL608617 0.79 KMO (0.73) KMOMKNK1MKNK2MEN1PSIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993019047-A1 TETRAHIDROPYRIDINYL (3/4) SUBSTITUED OXIMES HAVING SIGMA RECEPTOR AFFINITY AND THEIR USE IN THE TREATMENT OF CENTRAL NERVOUS SYSTEM CONDITIONS WARNER-LAMBERT COMPANY (US) 1993-09-30 WO disclosed
US-3991197-A ANALGESICS HOFFMANN-LA ROCHE INC. (US) 1976-11-09 US disclosed