SCHEMBL7365582

SCHEMBL7365582

CCCc1nn(C)c2c1N=C(c1sc(S(=O)(=O)N3CCN(CCO)CC3)cc1OCC)[N]C2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 19/20 0.46
PDE3B Q13370 3/20 0.46
PDE3A Q14432 3/20 0.46
PDE1A P54750 8/20 0.39
PDE1B Q01064 8/20 0.39
PDE1C Q14123 8/20 0.39
HDAC1 Q13547 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC2 Q92769 1/20 0.36
PDE2A O00408 1/20 0.35
ABCC4 O15439 1/20 0.35
ABCC5 O15440 1/20 0.35
PDE6D O43924 1/20 0.35
PDE8A O60658 1/20 0.35
PDE9A O76083 1/20 0.35
ABCB11 O95342 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
PDE6A P16499 1/20 0.35
PDE6G P18545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359421 0.91 PDE5A (0.42) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7426355 0.88 PDE5A (0.36) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7782809 0.78 PDE5A (0.55) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7402702 0.76 PDE5A (0.71) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL5795456 0.74 CA12 (0.59) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7449440 0.71 PDE5A (0.56) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7361790 0.69
SCHEMBL6624319 0.67 PDE5A (0.69) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL7431615 0.67 PDE5A (0.48) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL5076135 0.66 PDE5A (0.54) PDE5APDE3BPDE3APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001003644-A9 PYRAZOLOPYRIMIDINONE DERIVATIVES CONJUGATED TO THIOPHENE MOIETIES OR BENZO [FUSED] 5-MEMBERED HETEROCYCLES FOR ERECTILE DYSFUNCTION PICOWER INST MED RES (US) 2001-11-29 WO claimed