SCHEMBL7365919

SCHEMBL7365919

NC(=O)c1cc(O)ccc1C[CH]C(=O)N1CCC(CCCl)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
BTK Q06187 2/20 0.34
PARP14 Q460N5 2/20 0.34
TNKS O95271 1/20 0.33
PARP1 P09874 1/20 0.33
TEAD1 P28347 1/20 0.33
TEAD3 Q99594 1/20 0.33
CCR2 P41597 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MGLL Q99685 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364619 0.90 BTK (0.37) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7444511 0.76 PARP14 (0.36) BTKPARP14TNKSPARP1HTR2A
SCHEMBL4096182 0.76 HTR2A (0.40) BTKPARP14TNKSPARP1HTR2A
SCHEMBL3140703 0.73 PARP1 (0.43) BTKPARP14TNKSPARP1HTR2A
SCHEMBL5090081 0.71 LCK (0.40) KMT2APARP1ALDH1A1
SCHEMBL7369342 0.71 TEAD1 (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3127933 0.68 BCHE (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7363740 0.67 GRIN2D (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7365927 0.66 GRIN2D (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3140842 0.65 ALDH1A1 (0.35) BTKPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997046553-A1 THROMBIN INHIBITORS NOVARTIS AG (CH) 1997-12-11 WO disclosed