SCHEMBL7365960

SCHEMBL7365960

O=C(c1cccc(C=S)c1)c1cccnc1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.51
ALDH1A1 P00352 4/20 0.51
MAPT P10636 2/20 0.51
CYP3A4 P08684 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
BLM P54132 1/20 0.51
AGER Q15109 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
UNG P13051 1/20 0.40
GAA P10253 1/20 0.39
POLB P06746 1/20 0.38
NEK2 P51955 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.37
DHODH Q02127 3/20 0.37
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369369 0.89 ALDH1A1 (0.51) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL296670 0.79 KDM4E (0.69) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7366851 0.79 ALOX15 (0.56) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7366513 0.79 MAPT (0.56) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7366799 0.79 POLB (0.63) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL9375327 0.78 KDM4E (0.54) KDM4EALDH1A1MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL7853761 0.78 KDM4E (0.67) KDM4EALDH1A1MAPTCYP3A4ALOX15
Oxalic Acid SCHEMBL31550428 0.76 KDM4E (0.65) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7369163 0.76 ALDH1A1 (0.54) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL7370589 0.76 ALDH1A1 (0.55) KDM4EALDH1A1MAPTCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed