SCHEMBL7366105

SCHEMBL7366105

CCCCCC(=O)Nc1ccc(C(=O)Cl)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.63
THRB P10828 1/20 0.63
ALDH1A1 P00352 1/20 0.61
CA1 P00915 2/20 0.60
CA2 P00918 2/20 0.60
ENPP2 Q13822 1/20 0.57
DGAT2 Q96PD7 1/20 0.57
PSMB11 A5LHX3 1/20 0.57
PSMA7 O14818 1/20 0.57
PSMB1 P20618 1/20 0.57
PSMA1 P25786 1/20 0.57
PSMA2 P25787 1/20 0.57
PSMA3 P25788 1/20 0.57
PSMA4 P25789 1/20 0.57
PSMB8 P28062 1/20 0.57
PSMB9 P28065 1/20 0.57
PSMA5 P28066 1/20 0.57
PSMB4 P28070 1/20 0.57
PSMB6 P28072 1/20 0.57
PSMB5 P28074 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9510547 0.86 ENPP2 (0.71) THRATHRBALDH1A1CA1CA2
SCHEMBL675018 0.86 ENPP2 (0.71) THRATHRBALDH1A1CA1CA2
SCHEMBL9858666 0.86 ENPP2 (0.71) THRATHRBALDH1A1CA1CA2
SCHEMBL11801804 0.85 ALDH1A1 (0.68) THRATHRBALDH1A1CA1CA2
SCHEMBL11801797 0.85 THRA (0.65) THRATHRBALDH1A1CA1CA2
SCHEMBL76386 0.84 ALDH1A1 (0.66) THRATHRBALDH1A1CA1CA2
SCHEMBL7813320 0.84 ALDH1A1 (0.66) THRATHRBALDH1A1CA1CA2
SCHEMBL5215426 0.84 ALDH1A1 (0.66) THRATHRBALDH1A1CA1CA2
SCHEMBL21998909 0.84 ALDH1A1 (0.66) THRATHRBALDH1A1CA1CA2
SCHEMBL7829195 0.84 ALDH1A1 (0.66) THRATHRBALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804420-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed