SCHEMBL7366329

SCHEMBL7366329

COC(=O)c1c(C2CCN(c3ccncc3)CC2)ccc(N)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.44
CYP3A4 P08684 4/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP2C19 P33261 1/20 0.40
CYP2C9 P11712 3/20 0.39
CYP2D6 P10635 3/20 0.39
HRH3 Q9Y5N1 1/20 0.39
TSHR P16473 2/20 0.39
F10 P00742 6/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
F2 P00734 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
HTR4 Q13639 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5221896 0.70 HIF1A (0.41) HIF1ACYP3A4CYP2C9CYP2D6HRH3
SCHEMBL5759922 0.69 MAPT (0.62) HIF1ACYP3A4ALDH1A1CYP2C9CYP2D6
SCHEMBL31519913 0.68 ALDH1A1 (0.46) ALDH1A1TSHRKDM4EHPGD
SCHEMBL5222775 0.68 MEN1 (0.47) CYP3A4CYP2C19CYP2C9F10ITGB3
SCHEMBL5224718 0.67 HDAC3 (0.42) F10ITGB3ITGA2BHTR4
SCHEMBL5227299 0.67 HIF1A (0.50) HIF1ACYP3A4ALDH1A1CYP2C19CYP2C9
Hydrochloric Acid SCHEMBL5225043 0.67 HDAC3 (0.41) F10ITGB3ITGA2BHTR4
SCHEMBL5227295 0.66 HIF1A (0.49) HIF1ACYP3A4ALDH1A1CYP2C19CYP2C9
SCHEMBL31150607 0.66 FAAH (0.41) ALDH1A1TSHRKDM4ENPC1MAPT
SCHEMBL12426327 0.66 F10 (0.49) ALDH1A1F10HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019045-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2002-07-03 EP disclosed
EP-1019045-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-19 EP disclosed
WO-1999000128-A9 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 1999-08-05 WO disclosed
WO-1999000128-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed