SCHEMBL7366443

SCHEMBL7366443

O=C(O)CCNC(=O)NC(Cc1ccccc1)CP(=O)(O)O

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MME P08473 2/20 0.51
ACE P12821 2/20 0.51
ECE1 P42892 1/20 0.48
MMEL1 Q495T6 1/20 0.45
CCR3 P51677 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367862 0.86 MME (0.54) MMEACEECE1MMEL1
SCHEMBL9588091 0.82 MME (0.62) MMEACEECE1
SCHEMBL7370588 0.82 MME (0.59) MMEACE
SCHEMBL7318461 0.80 ACE (0.70) MMEACEECE1MMEL1
SCHEMBL7367811 0.80 ACE (0.70) MMEACEECE1MMEL1
SCHEMBL7367809 0.80 ACE (0.70) MMEACEECE1MMEL1
SCHEMBL7365324 0.79 MME (0.66) MMEACE
SCHEMBL7367162 0.78 NAALAD2 (0.58) MME
SCHEMBL7367157 0.78 NAALAD2 (0.58) MME
SCHEMBL10791111 0.78 ACE (0.68) MMEACEECE1MMEL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0117429-B1 PHOSPHOROUS CONTAINING COMPOUNDS AS INHIBITORS OF ENKEPHALINASES SCHERING CORPORATION (US) 1987-09-02 EP claimed
EP-0117429-A1 Phosphorous containing compounds as inhibitors of enkephalinases SCHERING CORPORATION (US) 1984-09-05 EP claimed
EP-0117429-B1 PHOSPHOROUS CONTAINING COMPOUNDS AS INHIBITORS OF ENKEPHALINASES SCHERING CORPORATION (US) 1987-09-02 EP disclosed
EP-0117429-A1 Phosphorous containing compounds as inhibitors of enkephalinases SCHERING CORPORATION (US) 1984-09-05 EP disclosed