SCHEMBL7366987

SCHEMBL7366987

CC(C)(C)OC(=O)NCCC(C(=O)c1oc(-c2ccccc2)nc1-c1ccccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.45
SKP1 P63208 2/20 0.45
SKP2 Q13309 2/20 0.45
S1PR1 P21453 1/20 0.42
ATR Q13535 1/20 0.41
IDO1 P14902 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.39
MALT1 Q9UDY8 1/20 0.39
GABRA5 P31644 1/20 0.39
NPSR1 Q6W5P4 4/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 2/20 0.38
BCHE P06276 1/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802903 0.77 CTSK (0.53) MEN1KMT2AALDH1A1CTSSCTSK
SCHEMBL4583816 0.76 MEN1 (0.54) IDO1MALT1NPSR1MEN1KMT2A
SCHEMBL6335913 0.76 CKS1B (0.43) CKS1BSKP1SKP2S1PR1ATR
SCHEMBL29182105 0.74 MEN1 (0.49) CKS1BSKP1SKP2S1PR1IDO1
SCHEMBL7049753 0.74 BCHE (0.41) S1PR1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL20014854 0.72 MTNR1A (0.61) IDO1MALT1MEN1KMT2ACTSS
SCHEMBL6676845 0.71 CYP1A2 (0.43) CKS1BSKP1SKP2IDO1MALT1
SCHEMBL14148637 0.70 KDR (0.53) CKS1BSKP1SKP2SMN1; SMN2MAPT
SCHEMBL16084764 0.70 RIPK1 (0.53) IDO1MALT1MEN1KMT2ABCHE
SCHEMBL1521024 0.70 RIPK1 (0.53) IDO1MALT1MEN1KMT2ABCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed