SCHEMBL7367074

SCHEMBL7367074

COC(=O)c1nnc(CBr)s1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.41
HSD17B10 Q99714 3/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 2/20 0.38
GLS O94925 1/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
TSHR P16473 2/20 0.35
KMT2A Q03164 2/20 0.35
RECQL P46063 1/20 0.35
LMNA P02545 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18352875 0.75 CES1 (0.42) CES1HSD17B10HTTALDH1A1MAPT
SCHEMBL22272749 0.75 POLB (0.62) CES1HSD17B10SMN1; SMN2ALDH1A1MAPT
SCHEMBL7453197 0.74 SMN1; SMN2 (0.43) CES1HSD17B10SMN1; SMN2ALDH1A1MAPT
SCHEMBL368639 0.72 HSD17B10 (0.50) CES1HSD17B10HTTSMN1; SMN2ALDH1A1
SCHEMBL27264408 0.72 TSHR (0.42) CES1HSD17B10HTTSMN1; SMN2ALDH1A1
SCHEMBL17967149 0.72 FFAR1 (0.48) CES1ALDH1A1KMT2ALMNAMEN1
SCHEMBL8356502 0.72 HSD17B10 (0.47) HSD17B10SMN1; SMN2ALDH1A1GLSMAPT
SCHEMBL25144949 0.71 ALDH1A1 (0.40) CES1HSD17B10SMN1; SMN2ALDH1A1MAPT
SCHEMBL19948875 0.70 ALDH1A1 (0.40) CES1HSD17B10SMN1; SMN2ALDH1A1MAPT
SCHEMBL9800508 0.69 ALDH1A1 (0.41) CES1HSD17B10SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691329-A Compounds containing basic and acidic termini useful as fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-25 US disclosed
US-5563158-A CARDIOVASCULAR DISORDERS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-08 US disclosed
WO-1995018111-A1 COMPOUNDS CONTAINING BASIC AND ACIDIC TERMINI USEFUL AS FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-07-06 WO disclosed