SCHEMBL7367363

SCHEMBL7367363

COC(=O)CC12CCN(CC1)C2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
TSHR P16473 3/20 0.34
HSD17B10 Q99714 1/20 0.32
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
GLA P06280 1/20 0.31
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367053 0.93 CHRM2 (0.34) TP53TSHRCHRM2CHRM4CHRM1
SCHEMBL9696852 0.81 KMT2A (0.44) TSHRMGAMGAASIMGAM2
SCHEMBL22784325 0.75 GRM1 (0.38) TSHRUSP2
Bromide SCHEMBL10316864 0.74 CTSK (0.31)
SCHEMBL7985447 0.72 CHRM2 (0.40) TSHRHSD17B10MGAMGAASI
SCHEMBL22784402 0.70
SCHEMBL2422852 0.69 KMT2A (0.42) TSHRMGAMGAASIMGAM2
SCHEMBL4493164 0.69 CHRM2 (0.37) CHRM2CHRM4CHRM1CHRM3
SCHEMBL22912579 0.69 CHRM2 (0.32) CHRM2CHRM4CHRM1CHRM3
SCHEMBL22784397 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625981-A1 AZABICYCLO COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-11-30 EP disclosed
WO-1993015080-A1 AZABICYCLO COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-08-05 WO disclosed