SCHEMBL7367369

SCHEMBL7367369

CON(C)C(=O)COc1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.52
TSHR P16473 1/20 0.52
SENP2 Q9HC62 1/20 0.49
SENP1 Q9P0U3 1/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
POLB P06746 3/20 0.48
RAB9A P51151 2/20 0.48
MAPT P10636 2/20 0.48
RECQL P46063 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TP53 P04637 4/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257484 0.81 KDM4E (0.50) HPGDMEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL22232434 0.80 MRGPRX4 (0.49) HPGDTSHRMEN1KMT2ASMN1; SMN2
SCHEMBL16382639 0.78 MEN1 (0.48) HPGDTSHRMEN1KMT2ASMN1; SMN2
SCHEMBL4842036 0.77 SMN1; SMN2 (0.63) MEN1KMT2ASMN1; SMN2RAB9AKDM4E
SCHEMBL5000478 0.77 LMNA (0.62) HPGDTSHRSENP2SENP1MEN1
SCHEMBL5523413 0.76 KMT2A (0.57) HPGDTSHRSENP2SENP1MEN1
SCHEMBL101520 0.74 PTGDR2 (0.68) HPGDTSHRMEN1KMT2ASMN1; SMN2
SCHEMBL3254718 0.74 MEN1 (0.58) HPGDTSHRSENP2SENP1MEN1
SCHEMBL2011265 0.74 USP2 (0.58) HPGDTSHRSENP2SENP1MEN1
SCHEMBL1515893 0.74 SIGMAR1 (0.47) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380218-B1 FOR THERAPY OF RESPIRATORY, ALLERGIC, AND INFLAMMATORY DISORDERS COMPRISING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ACUTE RESPIRATORY DISEASE SYNDROME, PULMONARY HYPERSENSITIVITY, AND ALLERGIC RHINITIS IN A MAMMAL PFIZER INC 2002-04-30 US disclosed
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed