SCHEMBL7367403

SCHEMBL7367403

CC(C)C[C@@H](C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCNCCO)N(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.51
CTSK P43235 5/20 0.51
CTSL P07711 3/20 0.49
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
CPA1 P15085 1/20 0.48
ACE2 Q9BYF1 1/20 0.48
MMP8 P22894 2/20 0.47
MMP9 P14780 1/20 0.47
PTPN1 P18031 1/20 0.45
NPC1 O15118 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PLG P00747 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44
IL1RN P18510 1/20 0.44
ERAP2 Q6P179 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190103 0.91 CTSS (0.47) CTSSCTSKCTSLMMEACE
SCHEMBL7340564 0.88 CTSS (0.52) CTSSCTSKCTSLMMEACE
SCHEMBL8210636 0.85 ACE (0.64) MMEACECPA1ACE2MMP8
SCHEMBL8210634 0.85 ACE (0.64) MMEACECPA1ACE2MMP8
SCHEMBL7408154 0.84 CTSS (0.54) CTSSCTSKCTSLMMEACE
SCHEMBL7406564 0.83 CTSS (0.48) CTSSCTSKCTSLMMEACE
SCHEMBL7398380 0.83 CTSS (0.53) CTSSCTSKCTSLNPC1RAB9A
SCHEMBL7409019 0.83 MME (0.54) MMEACECPA1ACE2MMP8
SCHEMBL7343773 0.82 CACNA1B (0.55) CTSSCTSKCTSLPTPN1
SCHEMBL7370652 0.82 TACR2 (0.61) MMP8MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed