SCHEMBL7367434

SCHEMBL7367434

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccc(OCC(=O)O)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 4/20 0.47
HPGD P15428 2/20 0.47
POLB P06746 1/20 0.47
NR1I2 O75469 1/20 0.47
LMNA P02545 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
HIF1A Q16665 2/20 0.45
TSHR P16473 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TP53 P04637 1/20 0.45
CYP2D6 P10635 1/20 0.45
NFKB1 P19838 1/20 0.45
THPO P40225 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358485 0.89 KDM4E (0.48) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL7356152 0.81 CACNA1F (0.62) POLBLMNACYP1A2CYP3A4CYP2C9
SCHEMBL7362882 0.81 NR1I2 (0.64) KDM4EALDH1A1HSD17B10HPGDNR1I2
SCHEMBL7358619 0.80 ADORA3 (0.60) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL3006534 0.78 KDM4E (0.66) KDM4EALDH1A1HSD17B10HPGDNR1I2
SCHEMBL7390505 0.77 MAPT (0.56) KDM4EHSD17B10POLBTSHR
SCHEMBL9500152 0.75 TSHR (0.51) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL29676206 0.74 NR1I2 (0.73) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL3034560 0.74 NR1I2 (0.73) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL7414856 0.73 NR1I2 (0.67) KDM4EALDH1A1HSD17B10HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378718-A Cardiovascular activity, hypotensive CEDONA PHARMACEUTICALS B.V. (NL) 1995-01-03 US disclosed
WO-1992002503-A1 NOVEL 1,4-DIHYDROPYRIDINE DERIVATIVES CEDONA PHARMACEUTICALS BV (NL) 1992-02-20 WO disclosed