SCHEMBL7367477

SCHEMBL7367477

COc1cccc(-c2nn3ccncc3c2-c2nnccc2S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
GAA P10253 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
AURKA O14965 1/20 0.37
PTGDR2 Q9Y5Y4 3/20 0.37
HTT P42858 2/20 0.37
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BRAF P15056 1/20 0.36
MAPK14 Q16539 1/20 0.36
CYP11B1 P15538 5/20 0.36
CYP11B2 P19099 4/20 0.36
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364012 0.85 PTGS2 (0.35) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL7367472 0.82 KDM4E (0.39) ALDH1A1GAAKDM4ECYP3A4HPGD
SCHEMBL7364009 0.68 LMNA (0.37) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL7373754 0.68 IGF1R (0.39) AURKAPTGDR2MAPK14
SCHEMBL5673928 0.67 MAPK14 (0.40) CYP3A4AURKAPTGDR2MAPK14CYP11B1
SCHEMBL6818747 0.66 AURKA (0.39) ALDH1A1GAAKDM4ECYP3A4HPGD
SCHEMBL5673943 0.63 KDR (0.42) CYP3A4MAPK14CYP11B1MEN1KMT2A
SCHEMBL3652098 0.63 BRAF (0.46) ALDH1A1GAAKDM4ECYP3A4HPGD
SCHEMBL5671102 0.62 MAPK14 (0.50) LMNANPSR1BRAFMAPK14
SCHEMBL28279253 0.62 DYRK1A (0.51) ALDH1A1GAAKDM4ECYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244669-A1 PYRAZOLOPYRAZINES AND THEIR USE AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-10-02 EP disclosed
WO-2001040230-A1 PYRAZOLOPYRAZINES AND THEIR USE AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-07 WO disclosed