SCHEMBL7367495

SCHEMBL7367495

CN(CCN(C)C(=O)OCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
F13A1 P00488 1/20 0.54
TGM2 P21980 1/20 0.54
TGM1 P22735 1/20 0.54
MAPT P10636 1/20 0.53
HPGD P15428 1/20 0.53
TDP1 Q9NUW8 2/20 0.52
MAPK1 P28482 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
KMT2A Q03164 1/20 0.52
HDAC1 Q13547 1/20 0.50
CCR6 P51684 1/20 0.50
PAX8 Q06710 1/20 0.50
SIGMAR1 Q99720 1/20 0.48
ABCB1 P08183 1/20 0.48
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31697957 0.95 ALDH1A1 (0.53) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL25978639 0.95 ALDH1A1 (0.53) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL17067258 0.93 ALDH1A1 (0.56) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL25787612 0.92 ALDH1A1 (0.50) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL553299 0.91 ALDH1A1 (0.53) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL2724661 0.91 ALDH1A1 (0.53) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL13181407 0.91 LTB4R (0.56) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL1329140 0.90 HDAC1 (0.52) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL164180 0.90 ALDH1A1 (0.51) ALDH1A1F13A1TGM2TGM1MAPT
SCHEMBL11622571 0.90 ALDH1A1 (0.51) ALDH1A1F13A1TGM2TGM1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5348953-A Elastase inhibitor MERCK & CO., INC. (US) 1994-09-20 US disclosed
EP-0525973-A2 Substituted azetidinones as anti-inflammatory and antidegenerative agents MERCK & CO. INC. (US) 1993-02-03 EP disclosed
WO-1993000332-A1 SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS MERCK & CO., INC. (US) 1993-01-07 WO disclosed