SCHEMBL7367613

SCHEMBL7367613

N#Cc1ccc2c(ccn2CCC(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.52
FFAR4 Q5NUL3 1/20 0.51
P2RX7 Q99572 1/20 0.49
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
TSHR P16473 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
GLA P06280 1/20 0.44
HTT P42858 1/20 0.44
CYP19A1 P11511 1/20 0.44
PRMT5 O14744 1/20 0.44
ITGB3 P05106 3/20 0.43
ITGAV P06756 3/20 0.43
ITGB5 P18084 2/20 0.43
ITGB1 P05556 1/20 0.43
ITGA5 P08648 1/20 0.43
LMNA P02545 1/20 0.42
RORC P51449 1/20 0.42
NPY5R Q15761 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413159 0.92 FFAR4 (0.55) KMOFFAR4P2RX7KDM4EALDH1A1
SCHEMBL5487411 0.89 P2RX7 (0.54) KMOFFAR4P2RX7KDM4EALDH1A1
SCHEMBL3465527 0.85 KMT2A (0.55) FFAR4P2RX7KDM4EALDH1A1TSHR
SCHEMBL403709 0.82 TNF (0.49) FFAR4P2RX7CYP19A1PRMT5RORC
SCHEMBL17242442 0.79 P2RX7 (0.54) FFAR4P2RX7KDM4EALDH1A1TSHR
SCHEMBL28315634 0.79 P2RX7 (0.50) P2RX7CYP19A1PRMT5RORCNPY5R
SCHEMBL30041872 0.79 PRMT5 (0.49) FFAR4P2RX7KDM4EALDH1A1TSHR
SCHEMBL17242289 0.78 P2RX7 (0.56) FFAR4P2RX7KDM4EALDH1A1TSHR
SCHEMBL4327022 0.78 HDAC1 (0.53) P2RX7KDM4EALDH1A1TSHRHSD17B10
SCHEMBL1576323 0.78 KMO (0.78) KMOITGB3ITGAVITGB5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043257-A ANTICOAGULANT; PYRIDINE SUBSTITUTED INDAZOLE COMPOUND E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-03-28 US disclosed
EP-0960102-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN Du Pont Pharmaceuticals Company (US) 1999-12-01 EP disclosed
US-5886191-A ANTICOAGULANTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-23 US disclosed
WO-1998001428-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN DU PONT PHARMACEUTICALS COMPANY (US) 1998-01-15 WO disclosed