SCHEMBL7367934

SCHEMBL7367934

CC(C)C[C@H](NC1CCOCC1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCNCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 7/20 0.51
CTSS P25774 7/20 0.49
CTSK P43235 6/20 0.49
CTSL P07711 3/20 0.49
PLG P00747 1/20 0.48
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
YAP1 P46937 1/20 0.45
PTPN1 P18031 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370096 0.88 TACR2 (0.60) TACR2
SCHEMBL7408901 0.87 TACR2 (0.54) TACR2CTSSYAP1
SCHEMBL7367334 0.85 CACNA1B (0.54) TACR2CTSSYAP1PTPN1
SCHEMBL8207767 0.83 REN (0.48) TACR2CTSSCTSKCTSLYAP1
SCHEMBL7368981 0.83 CACNA1B (0.58) TACR2CTSSCTSK
SCHEMBL7402583 0.83 TACR2 (0.54) TACR2CTSSCTSK
SCHEMBL7371474 0.83 YAP1 (0.53) CTSSCTSKCTSLYAP1PTPN1
SCHEMBL7371480 0.83 YAP1 (0.53) CTSSCTSKCTSLYAP1PTPN1
SCHEMBL8194350 0.83 IL1RN (0.48) TACR2CTSSCTSKCTSLYAP1
SCHEMBL7371242 0.83 CACNA1B (0.61) CTSSYAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed