SCHEMBL7367334

SCHEMBL7367334

CC(C)C[C@H](NC1CCOCC1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.54
YAP1 P46937 3/20 0.49
REN P00797 1/20 0.48
IL1RN P18510 1/20 0.48
ERAP2 Q6P179 1/20 0.48
ERAP1 Q9NZ08 1/20 0.48
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
CPA1 P15085 1/20 0.48
ACE2 Q9BYF1 1/20 0.48
PTPN1 P18031 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
PSMB11 A5LHX3 2/20 0.45
PSMA7 O14818 2/20 0.45
PSMB1 P20618 2/20 0.45
PSMA1 P25786 2/20 0.45
PSMA2 P25787 2/20 0.45
PSMA3 P25788 2/20 0.45
PSMA4 P25789 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8207767 0.93 REN (0.48) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL8180144 0.90 YAP1 (0.45) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL7371474 0.89 YAP1 (0.53) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL7371480 0.89 YAP1 (0.53) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL8194350 0.85 IL1RN (0.48) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL7367934 0.85 TACR2 (0.51) YAP1PTPN1TACR2CTSS
SCHEMBL7371242 0.85 CACNA1B (0.61) CACNA1BYAP1RENPSMB11PSMA7
SCHEMBL7370096 0.85 TACR2 (0.60) MMP9MMP8PSMB11PSMA7PSMB1
SCHEMBL7399618 0.85 CACNA1B (0.52) CACNA1BYAP1RENIL1RNERAP2
SCHEMBL7364989 0.84 MME (0.56) CACNA1BYAP1RENIL1RNERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed