SCHEMBL7368142

SCHEMBL7368142

Nc1cnc2c(n1)CCN(Cc1ccccc1)CC2

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
SIGMAR1 Q99720 2/20 0.49
HRH3 Q9Y5N1 1/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
GAA P10253 1/20 0.48
DHFR P00374 1/20 0.46
DRD2 P14416 1/20 0.46
KCNH2 Q12809 1/20 0.46
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.45
DRD4 P21917 1/20 0.45
ALDH1A1 P00352 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
MC4R P32245 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11078869 0.90 MEN1 (0.54) MEN1KMT2AHRH3NPC1RAB9A
Hydrochloric Acid SCHEMBL11072223 0.90 KMT2A (0.54) MEN1KMT2AHRH3NPC1RAB9A
SCHEMBL11069076 0.87 HSP90AB1 (0.49) MEN1KMT2ASIGMAR1DRD2KCNH2
Hydrochloric Acid SCHEMBL11068135 0.85 NOS3 (0.49) SIGMAR1HRH3DRD2
SCHEMBL30063704 0.84 SIGMAR1 (0.50) MEN1KMT2ASIGMAR1NPC1RAB9A
Hydrochloric Acid SCHEMBL11068298 0.82 SIGMAR1 (0.53) MEN1KMT2ASIGMAR1LMNAALDH1A1
SCHEMBL30063685 0.82 SIGMAR1 (0.49) MEN1KMT2ASIGMAR1NPC1RAB9A
SCHEMBL2580524 0.79 MEN1 (0.56) MEN1KMT2ASIGMAR1NPC1RAB9A
SCHEMBL11069340 0.79 SIGMAR1 (0.61) MEN1KMT2ASIGMAR1HRH3NPC1
SCHEMBL30063678 0.79 C5AR1 (0.51) MEN1KMT2ASIGMAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048702-A1 BENZAZEPINE DERIVATIVES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1997-12-24 WO disclosed
US-4486433-A SLOWING HEART RATE DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-12-04 US disclosed
US-4409220-A Fused-ring amino-pyrazines as bradycardiac agents DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-10-11 US disclosed
EP-0047412-A1 Pyrazines, their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1982-03-17 EP disclosed