SCHEMBL7368640

SCHEMBL7368640

O=C(CCc1ccccc1)c1cccnc1Oc1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
MAPK8 P45983 1/20 0.53
TDP1 Q9NUW8 1/20 0.49
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TBXAS1 P24557 1/20 0.44
CES1 P23141 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402170 0.90 KMT2A (0.48) ALDH1A1MAPK8
SCHEMBL7403292 0.86 ALDH1A1 (0.42) ALDH1A1MAPK8TDP1
SCHEMBL7369624 0.83 KMT2A (0.57) ALDH1A1MAPK8TDP1
SCHEMBL5216488 0.80 TDP1 (0.56) ALDH1A1MAPK8TDP1CYP3A4
SCHEMBL5218853 0.79 ALDH1A1 (0.54) ALDH1A1MAPK8TDP1
SCHEMBL7675867 0.79 ALDH1A1 (0.52) ALDH1A1MAPK8TDP1
SCHEMBL7677170 0.78 MAPK8 (0.54) ALDH1A1MAPK8TDP1
SCHEMBL7370595 0.78 MAPK8 (0.50) ALDH1A1MAPK8TDP1TBXAS1
SCHEMBL7677512 0.78 KMT2A (0.53) ALDH1A1MAPK8
SCHEMBL7694995 0.76 TDP1 (0.55) ALDH1A1MAPK8TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380218-B1 FOR THERAPY OF RESPIRATORY, ALLERGIC, AND INFLAMMATORY DISORDERS COMPRISING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ACUTE RESPIRATORY DISEASE SYNDROME, PULMONARY HYPERSENSITIVITY, AND ALLERGIC RHINITIS IN A MAMMAL PFIZER INC 2002-04-30 US disclosed
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed