SCHEMBL7368764

SCHEMBL7368764

CCOC(=O)CCCOc1ccccc1N(C)C(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
KMT2A Q03164 3/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
POLB P06746 2/20 0.44
MAPT P10636 9/20 0.44
LMNA P02545 3/20 0.43
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 4/20 0.42
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
GLA P06280 1/20 0.40
NPC1 O15118 1/20 0.40
S1PR4 O95977 1/20 0.40
ITGA4 P13612 1/20 0.40
HPGD P15428 1/20 0.40
S1PR1 P21453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337134 0.96 ALDH1A1 (0.49) ALDH1A1KMT2AMAPK1TDP1POLB
SCHEMBL7377964 0.89 POLB (0.56) ALDH1A1KMT2AMAPK1POLBMAPT
SCHEMBL7374177 0.84 CRHBP (0.44) ALDH1A1KMT2AMAPTLMNAL3MBTL1
SCHEMBL7373301 0.84 MAPK1 (0.45) ALDH1A1KMT2AMAPK1TDP1POLB
SCHEMBL7368736 0.82 KMT2A (0.46) ALDH1A1KMT2AMAPK1TDP1MAPT
SCHEMBL7368292 0.82 ALDH1A1 (0.44) ALDH1A1KMT2AMAPK1TDP1MAPT
SCHEMBL7368288 0.82 ALDH1A1 (0.44) ALDH1A1KMT2AMAPK1TDP1MAPT
SCHEMBL7376305 0.81 MAPT (0.48) ALDH1A1KMT2AMAPK1TDP1POLB
SCHEMBL7340316 0.81 MAPT (0.40) ALDH1A1KMT2ATDP1MAPTLMNA
SCHEMBL7376368 0.81 ALDH1A1 (0.48) ALDH1A1KMT2AMAPK1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed