SCHEMBL7368288

SCHEMBL7368288

CCOC(=O)CCCO/N=C/c1ccccc1N(C)C(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
KMT2A Q03164 5/20 0.44
TDP1 Q9NUW8 2/20 0.44
MAPK1 P28482 2/20 0.44
MAPT P10636 8/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
MEN1 O00255 3/20 0.36
PTPN1 P18031 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
MAOB P27338 1/20 0.36
TBXAS1 P24557 2/20 0.36
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368292 1.00 ALDH1A1 (0.44) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7370181 0.87 L3MBTL1 (0.38) ALDH1A1TDP1MAPK1LMNAL3MBTL1
SCHEMBL7368764 0.82 ALDH1A1 (0.46) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7368291 0.82 ALDH1A1 (0.43) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7377424 0.81 SNCA (0.51) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7377419 0.81 SNCA (0.51) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7337134 0.81 ALDH1A1 (0.49) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7373216 0.79 KMT2A (0.53) ALDH1A1KMT2ATDP1MAPK1MAPT
SCHEMBL7378630 0.78 AVPR2 (0.41) ALDH1A1KMT2AMAPK1MAPTLMNA
SCHEMBL7378634 0.78 AVPR2 (0.41) ALDH1A1KMT2AMAPK1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed