SCHEMBL7368873

SCHEMBL7368873

CCOC(=O)C1=C(CSC2(OC)CCCCC2)NC(C)=C(C(=O)OC)C1c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.49
CACNA1B Q00975 6/20 0.49
HIF1A Q16665 5/20 0.49
CYP2C9 P11712 5/20 0.49
MEN1 O00255 4/20 0.49
CYP1A2 P05177 4/20 0.49
CYP3A4 P08684 4/20 0.49
CYP2C19 P33261 4/20 0.49
KMT2A Q03164 4/20 0.49
MAPT P10636 3/20 0.49
LMNA P02545 2/20 0.49
CYP2D6 P10635 2/20 0.49
TSHR P16473 2/20 0.49
NFKB1 P19838 2/20 0.49
THPO P40225 2/20 0.49
POLB P06746 1/20 0.49
MAPK1 P28482 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49
ACHE P22303 1/20 0.45
KDM4E B2RXH2 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9501260 0.85 ADORA3 (0.57) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL7419122 0.81 ADORA3 (0.53) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL9502243 0.81 ADORA3 (0.73) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL7471880 0.81 ADORA3 (0.51) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL9669318 0.79 ADORA3 (0.50) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL7318265 0.78 CACNA1B (0.51) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL9513394 0.77 ABCC1 (0.58) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL11522715 0.77 ABCC1 (0.58) ADORA3CACNA1BHIF1ACYP2C9MEN1
SCHEMBL7318260 0.77 CACNA1B (0.52) ADORA3CACNA1BCACNA1FCACNA1DCACNA1S
SCHEMBL7316147 0.77 ADORA3 (0.53) ADORA3CACNA1BHIF1ACYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4971984-A Cardiovascular disorders, hypotensive agints BEEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1990-11-20 US disclosed
EP-0271059-A1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1988-06-15 EP disclosed