SCHEMBL7368963

SCHEMBL7368963

CC(C)(NC(=O)[CH]Cc1ccc(NCc2ccccc2)cc1)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.46
FFAR4 Q5NUL3 2/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
HTT P42858 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
MAPK1 P28482 1/20 0.42
GFER P55789 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 2/20 0.41
MRGPRX1 Q96LB2 1/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860635 0.80 KDM4E (0.49) HTTMAPTMEN1KMT2AALDH1A1
SCHEMBL7374110 0.79 EPHX2 (0.38) CA1CA2MAPTGFERALDH1A1
SCHEMBL27519262 0.74 FFAR1 (0.52) FFAR1FFAR4CA1CA2HTT
SCHEMBL7365531 0.73 ALDH1A1 (0.44) HTTGAAMAPTMEN1KMT2A
SCHEMBL7368965 0.71 FFAR1 (0.49) FFAR1FFAR4CA1CA2HTT
SCHEMBL7372533 0.71 SPHK1 (0.38) MAPTALOX15MAPK1HIF1AALDH1A1
N-Benzylaniline SCHEMBL28146501 0.70 FFAR1 (0.62) FFAR1FFAR4CA1CA2HTT
SCHEMBL6962941 0.70 FFAR1 (0.64) FFAR1FFAR4CA1CA2HTT
SCHEMBL2850028 0.69 RIPK1 (0.49) CA1GAAMAPTMEN1KMT2A
SCHEMBL7386531 0.69 FFAR1 (0.56) FFAR1FFAR4CA1CA2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed