SCHEMBL7369209

SCHEMBL7369209

NC(=O)c1cc(Cl)cc([N+](=O)[O-])c1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 1/20 0.46
CYP3A4 P08684 2/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
PARP1 P09874 1/20 0.42
KCNMA1 Q12791 1/20 0.40
VCAM1 P19320 1/20 0.40
BCL2L1 Q07817 1/20 0.40
TTR P02766 1/20 0.40
FLT1 P17948 1/20 0.38
FLT4 P35916 1/20 0.38
KDR P35968 1/20 0.38
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6121980 0.84 ALDH1A1 (0.47) ALDH1A1LMNAKMT2ATSHRCYP3A4
SCHEMBL630835 0.83 ALDH1A1 (0.68) ALDH1A1LMNAKMT2ACYP3A4MAPT
SCHEMBL14775885 0.83 TTR (0.50) ALDH1A1LMNAKMT2ACYP3A4MAPT
SCHEMBL31374314 0.83 TTR (0.50) ALDH1A1LMNAKMT2ACYP3A4MAPT
SCHEMBL7095093 0.83 ALDH1A1 (0.48) ALDH1A1LMNAKMT2ATSHRCYP3A4
SCHEMBL8842559 0.81 ALDH1A1 (0.47) ALDH1A1LMNAKMT2ACYP3A4MAPT
SCHEMBL11800281 0.79 TSHR (0.62) ALDH1A1LMNAKMT2ATSHRCYP3A4
SCHEMBL31218397 0.78 LMNA (0.47) ALDH1A1LMNAKMT2AMAPTPOLB
SCHEMBL6896167 0.77 HPGD (0.56) ALDH1A1LMNAKMT2ATSHRCYP3A4
SCHEMBL30176207 0.77 HPGD (0.56) ALDH1A1LMNAKMT2ATSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1085871-A4 QUINAZOLINONE INHIBITORS OF cGMP PHOSPHODIESTERASE BRISTOL MYERS SQUIBB CO (US) 2001-10-04 EP disclosed
EP-1085871-A1 QUINAZOLINONE INHIBITORS OF cGMP PHOSPHODIESTERASE BRISTOL-MYERS SQUIBB COMPANY (US) 2001-03-28 EP disclosed
WO-1999064004-A1 QUINAZOLINONE INHIBITORS OF cGMP PHOSPHODIESTERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-12-16 WO disclosed