SCHEMBL7369535

SCHEMBL7369535

O=C(CBr)C1(c2cccc(Cl)c2)CCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.44
SLC6A3 Q01959 4/20 0.44
CCR2 P41597 1/20 0.43
SLC6A2 P23975 2/20 0.41
HSD11B1 P28845 1/20 0.41
EP300 Q09472 3/20 0.41
CREBBP Q92793 3/20 0.41
IDO1 P14902 2/20 0.40
KCNH2 Q12809 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
HTR2C P28335 2/20 0.38
HDAC4 P56524 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2B P41595 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DPP4 P27487 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9466663 0.81 AKR1C1 (0.59) SLC6A4SLC6A3CCR2SLC6A2HSD11B1
SCHEMBL1769960 0.81 HDAC4 (0.54) HSD11B1HDAC4HDAC1
SCHEMBL16507538 0.80 AKR1C1 (0.58) HSD11B1HDAC4MEN1KMT2AAKR1C1
SCHEMBL7047849 0.80 SLC6A3 (0.47) SLC6A4SLC6A3CCR2SLC6A2
SCHEMBL7369115 0.80 CCR2 (0.49) SLC6A4SLC6A3CCR2SLC6A2HSD11B1
SCHEMBL4446356 0.80 SLC6A4 (0.44) SLC6A4SLC6A3CCR2SLC6A2HSD11B1
SCHEMBL18742689 0.80 LMNA (0.48) SLC6A4SLC6A3CCR2SLC6A2HSD11B1
SCHEMBL16523531 0.79 MEN1 (0.45) SLC6A4SLC6A3HSD11B1EP300CREBBP
SCHEMBL16521043 0.79 EPHX2 (0.55) SLC6A4SLC6A3SLC6A2HSD11B1EP300
SCHEMBL28595250 0.78 SLC6A4 (0.49) SLC6A4SLC6A3CCR2SLC6A2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715620-B1 1-ARYLCYCLOALKYL SULPHIDES, SULPHOXIDES AND SULPHONES FOR THE TREATMENT OF DEPRESSION, ANXIETY AND PARKINSON'S DISEASE KNOLL AG (DE) 1998-10-28 EP disclosed
US-5652271-A ANTIDEPRESSANTS, NERVOUS SYSTEM DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1997-07-29 US disclosed
EP-0715620-A1 1-ARYLCYCLOALKYL SULPHIDES, SULPHOXIDES AND SULPHONES FOR THE TREATMENT OF DEPRESSION, ANXIETY AND PARKINSON'S DISEASE Knoll AG (DE) 1996-06-12 EP disclosed
WO-1994026704-A1 1-ARYLCYCLOALKYL SULPHIDES, SULPHOXIDES AND SULPHONES FOR THE TREATMENT OF DEPRESSION, ANXIETY AND PARKINSON'S DISEASE THE BOOTS COMPANY PLC (GB) 1994-11-24 WO disclosed