SCHEMBL7369869

SCHEMBL7369869

C[C@@H](c1ccc(N)cc1)N(C)C(=O)OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.50
ALOX5 P09917 1/20 0.48
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.44
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371515 0.89 ABCB1 (0.49) ABCB1ALOX5MEN1LMNAKMT2A
SCHEMBL7367400 0.82 ALDH1A1 (0.47) ABCB1MEN1KMT2AALDH1A1
SCHEMBL1460239 0.80 ABCB1 (0.53) ABCB1MEN1KMT2AALDH1A1CTSL
SCHEMBL8276259 0.79 ABCB1 (0.56) ABCB1LMNAKMT2AALDH1A1CTSL
SCHEMBL21952369 0.79 ABCB1 (0.44) ABCB1MEN1LMNAKMT2AALDH1A1
SCHEMBL20004309 0.79 ALDH1A1 (0.50) ALOX5MEN1LMNAKMT2AALDH1A1
SCHEMBL5149951 0.78 ABCB1 (0.58) ABCB1LMNAKMT2AALDH1A1CTSL
SCHEMBL19754815 0.78 ABCB1 (0.49) ABCB1ALOX5MEN1LMNAKMT2A
SCHEMBL23220190 0.77 ABCB1 (0.42) ABCB1MEN1LMNAKMT2AALDH1A1
SCHEMBL30191411 0.77 ABCB1 (0.51) ABCB1KMT2AALDH1A1CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952321-A Substituted azetidinones as anti-inflammatory and antidegenerative agents MERCK & CO., INC. (US) 1999-09-14 US disclosed
EP-0666846-A4 1995-09-20 EP disclosed
EP-0666846-A1 NEW SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS MERCK & CO. INC. (US) 1995-08-16 EP disclosed
WO-1994010143-A1 NEW SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS MERCK & CO., INC. (US) 1994-05-11 WO disclosed