SCHEMBL7370236

SCHEMBL7370236

O=C[C@@H]1CSNC1C(=O)C=Cc1ccc(OCCCCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.48
S1PR3 Q99500 5/20 0.47
HPGD P15428 2/20 0.46
PPARA Q07869 2/20 0.43
FFAR1 O14842 1/20 0.43
PPARG P37231 1/20 0.41
CYSLTR2 Q9NS75 2/20 0.41
CYSLTR1 Q9Y271 2/20 0.41
S1PR5 Q9H228 1/20 0.41
GRIK2 Q13002 1/20 0.41
GSK3B P49841 1/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375337 0.90 HDAC1 (0.42) S1PR1S1PR3CYSLTR2CYSLTR1
SCHEMBL451122 0.75 S1PR1 (0.61) S1PR1S1PR3HPGDPPARAFFAR1
SCHEMBL451121 0.75 S1PR1 (0.61) S1PR1S1PR3HPGDPPARAFFAR1
SCHEMBL7370241 0.74 S1PR1 (0.48) S1PR1S1PR3HPGDPPARAFFAR1
SCHEMBL7370240 0.74 S1PR1 (0.48) S1PR1S1PR3HPGDPPARAFFAR1
SCHEMBL7366401 0.73 HDAC1 (0.43) HPGD
SCHEMBL7372051 0.70 HDAC1 (0.39) HPGD
SCHEMBL4657194 0.69 LMNA (0.61) S1PR1S1PR3PPARAFFAR1GSK3B
SCHEMBL4657195 0.69 LMNA (0.61) S1PR1S1PR3PPARAFFAR1GSK3B
SCHEMBL3083583 0.68 FFAR1 (0.60) S1PR1S1PR3HPGDFFAR1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805796-A1 CELL ADHESION INHIBITORS BIOGEN, INC. (US) 1997-11-12 EP claimed
EP-0461677-B1 Novel thiazolidine derivatives ONO PHARMACEUTICAL CO (JP) 1997-04-16 EP claimed
WO-1996022966-A1 CELL ADHESION INHIBITORS BIOGEN, INC. (US) 1996-08-01 WO claimed
EP-0461677-A1 Novel thiazolidine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1991-12-18 EP claimed
US-4857537-A PREVENTING AMNESIA ONO PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US claimed
EP-0280956-A1 Thiazolidine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1988-09-07 EP claimed
EP-0804435-A1 NOVEL IMIDAZOLE DERIVATIVES, METHOD FOR PREPARING SAME, NOVEL INTERMEDIATES THUS OBTAINED, MEDICINAL APPLICATIONS OF SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ROUSSEL UCLAF (FR) 1997-11-05 EP disclosed
WO-1996004275-A1 NOVEL IMIDAZOLE DERIVATIVES, METHOD FOR PREPARING SAME, NOVEL INTERMEDIATES THUS OBTAINED, MEDICINAL APPLICATIONS OF SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ROUSSEL UCLAF (FR) 1996-02-15 WO disclosed