SCHEMBL7370769

SCHEMBL7370769

COc1ccc(/C=C/C(=O)O)c(CN(CC(F)(F)F)C(=O)OC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.43
PTGER3 P43115 1/20 0.43
PTGER2 P43116 1/20 0.43
THRB P10828 1/20 0.38
ATM Q13315 1/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LY96 Q9Y6Y9 1/20 0.36
KEAP1 Q14145 2/20 0.35
NFE2L2 Q16236 2/20 0.35
JUN P05412 1/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370771 1.00 PTGER4 (0.43) PTGER4PTGER3PTGER2THRBATM
SCHEMBL6418150 0.91 LY96 (0.38) MAPTALDH1A1MEN1KMT2ACYP1A1
SCHEMBL6418148 0.91 LY96 (0.38) MAPTALDH1A1MEN1KMT2ACYP1A1
SCHEMBL6418683 0.82 SSTR4 (0.39) ALDH1A1MEN1KMT2A
SCHEMBL4639106 0.82 ALDH1A1 (0.34) THRBALDH1A1MEN1KMT2ANPC1
SCHEMBL4639101 0.82 ALDH1A1 (0.34) THRBALDH1A1MEN1KMT2ANPC1
SCHEMBL6418121 0.81 POLB (0.49) ALDH1A1KEAP1NFE2L2
SCHEMBL6420626 0.78 POLB (0.38) MAPTALDH1A1KMT2A
SCHEMBL7450078 0.78 MTNR1A (0.46) ALDH1A1NPC1RAB9A
SCHEMBL4638135 0.77 CYP1A2 (0.39) ALDH1A1KMT2AKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957917-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-05-15 EP disclosed
EP-0957917-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-24 EP disclosed
WO-1998014192-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-04-09 WO disclosed