SCHEMBL7370870

SCHEMBL7370870

O=C(CNC(=O)c1cccc(NC(=O)NCc2ccccn2)c1)NC(Cc1cccnc1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
TSHR P16473 2/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
ALOX15 P16050 1/20 0.52
GPR132 Q9UNW8 5/20 0.49
CMKLR2 P46091 1/20 0.49
CMKLR1 Q99788 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
KMT2A Q03164 1/20 0.48
NAMPT P43490 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778227 0.92 TSHR (0.58) SMN1; SMN2TSHRNPC1RAB9AGPR132
SCHEMBL7375033 0.90 SMN1; SMN2 (0.52) SMN1; SMN2TSHRNPC1RAB9AALOX15
SCHEMBL7337671 0.89 GPR132 (0.54) SMN1; SMN2TSHRGPR132CMKLR2CMKLR1
SCHEMBL7836171 0.88 TSHR (0.56) SMN1; SMN2TSHRNPC1GPR132CMKLR2
SCHEMBL7834296 0.86 NPC1 (0.55) SMN1; SMN2TSHRNPC1RAB9AGPR132
SCHEMBL7349960 0.85 GPR132 (0.53) SMN1; SMN2TSHRGPR132CMKLR2CMKLR1
SCHEMBL7341632 0.85 TSHR (0.49) SMN1; SMN2TSHRNPC1GPR132CMKLR2
SCHEMBL7834945 0.83 GPR132 (0.52) TSHRGPR132CMKLR2CMKLR1
SCHEMBL7349051 0.83 GPR132 (0.55) TSHRGPR132CMKLR2CMKLR1
SCHEMBL7823711 0.83 GPR139 (0.51) TSHRGPR132CMKLR2CMKLR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed