SCHEMBL7371577

SCHEMBL7371577

NCCCCc1nnc(C(=O)NCCC(=O)ONC(=O)OCc2ccccc2)s1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GLS O94925 9/20 0.46
FFAR1 O14842 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
HTT P42858 1/20 0.39
PRSS1 P07477 4/20 0.39
PRSS2 P07478 4/20 0.39
PRSS3 P35030 4/20 0.39
TPSAB1 Q15661 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371601 0.80 ITGB3 (0.51) GLSPRSS1PRSS2PRSS3TPSAB1
SCHEMBL7371595 0.80 ITGB3 (0.51) GLSPRSS1PRSS2PRSS3TPSAB1
SCHEMBL7371589 0.77 GLS (0.47) GLSFFAR1SMN1; SMN2PRSS1PRSS2
SCHEMBL8176914 0.76 SYK (0.44) GLSPRSS1PRSS2PRSS3TPSAB1
SCHEMBL8176909 0.76 SYK (0.44) GLSPRSS1PRSS2PRSS3TPSAB1
SCHEMBL7376134 0.73 CA12 (0.56) SMN1; SMN2HTT
SCHEMBL15724934 0.71 GLS (0.65) GLSFFAR1
SCHEMBL7415486 0.71 CA12 (0.56) SMN1; SMN2HTT
SCHEMBL27346972 0.71 CA12 (0.59) SMN1; SMN2HTT
SCHEMBL7105678 0.70 TDP1 (0.57) SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP disclosed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO disclosed