SCHEMBL7371601

SCHEMBL7371601

NCCCCc1nnc(C(=O)NC[C@H](NC(=O)OCc2ccccc2)C(=O)O)s1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.51
ITGA2B P08514 12/20 0.51
ITGAV P06756 9/20 0.51
GLS O94925 3/20 0.46
PRSS1 P07477 2/20 0.44
PRSS2 P07478 2/20 0.44
PRSS3 P35030 2/20 0.44
TPSAB1 Q15661 2/20 0.44
ECE1 P42892 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371595 1.00 ITGB3 (0.51) ITGB3ITGA2BITGAVGLSPRSS1
SCHEMBL8176909 0.90 SYK (0.44) ITGB3ITGA2BITGAVGLSPRSS1
SCHEMBL8176914 0.90 SYK (0.44) ITGB3ITGA2BITGAVGLSPRSS1
SCHEMBL8177114 0.85 ITGB3 (0.61) ITGB3ITGA2BITGAVGLS
SCHEMBL8177121 0.85 ITGB3 (0.61) ITGB3ITGA2BITGAVGLS
SCHEMBL7371589 0.84 GLS (0.47) ITGB3ITGA2BGLSPRSS1PRSS2
SCHEMBL8177327 0.82 ITGB3 (0.60) ITGB3ITGA2BITGAV
SCHEMBL8177321 0.81 ITGB3 (0.42) ITGB3ITGA2BITGAVGLS
SCHEMBL7371577 0.80 GLS (0.46) GLSPRSS1PRSS2PRSS3TPSAB1
SCHEMBL8176780 0.77 SYK (0.42) ITGB3ITGA2BITGAVGLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP disclosed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO disclosed