SCHEMBL7375133

SCHEMBL7375133

N#Cc1cc(C#N)cc(O[CH]Cc2cccnc2)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.42
RORC P51449 1/20 0.40
AR P10275 1/20 0.40
CYP11B1 P15538 5/20 0.40
VNN1 O95497 1/20 0.40
CYP11B2 P19099 5/20 0.40
CYP17A1 P05093 1/20 0.40
ALDH1A1 P00352 4/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2C19 P33261 3/20 0.37
HSD17B10 Q99714 3/20 0.37
CLK4 Q9HAZ1 3/20 0.37
ALOX15 P16050 2/20 0.37
MAPK1 P28482 2/20 0.37
TSHR P16473 1/20 0.37
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380196 0.78 MAPT (0.43) ALDH1A1CYP1A2
SCHEMBL7379186 0.77 LTA4H (0.45) CYP11B1CYP11B2ALDH1A1CYP1A2CYP3A4
SCHEMBL6742580 0.75 KDM4E (0.43) CYP11B1VNN1CYP11B2HSD17B10
SCHEMBL7378072 0.71 AR (0.42) CYP19A1ARCYP11B1VNN1CYP11B2
SCHEMBL7382349 0.71 VNN1 (0.39) CYP19A1ARCYP11B1VNN1CYP11B2
SCHEMBL23218256 0.70 CYP11B1 (0.50) CYP19A1CYP11B1CYP11B2ALDH1A1HSD17B10
SCHEMBL29593169 0.70 CYP11B1 (0.50) CYP19A1CYP11B1CYP11B2ALDH1A1HSD17B10
SCHEMBL6629615 0.69 CHRNB2 (0.48) ALDH1A1CYP1A2
SCHEMBL10474110 0.69 TDP1 (0.48)
SCHEMBL18002080 0.68 CYP11B1 (0.48) CYP11B1CYP11B2CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed