SCHEMBL7375164

SCHEMBL7375164

CN(C(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
ATM Q13315 1/20 0.46
CES1 P23141 2/20 0.44
CES2 O00748 1/20 0.44
ALDH1A1 P00352 3/20 0.44
GPBAR1 Q8TDU6 4/20 0.44
MAPK1 P28482 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
RORC P51449 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375065 0.82 CRHBP (0.52) CRHBPCRHR2ATMCES1CES2
SCHEMBL7371730 0.81 CRHBP (0.51) CRHBPCRHR2ATMCES1CES2
SCHEMBL7366943 0.81 GPBAR1 (0.44) GPBAR1
SCHEMBL10373835 0.81 ATM (0.54) CRHBPCRHR2ATMCES1CES2
SCHEMBL7375141 0.80 CRHBP (0.50) CRHBPCRHR2ATMCES1CES2
SCHEMBL30981379 0.80 CRHBP (0.50) CRHBPCRHR2ATMCES1CES2
SCHEMBL7368622 0.78 MAPK1 (0.53) CRHBPCRHR2ATMCES1CES2
SCHEMBL8812280 0.77 ALDH1A1 (0.53) CRHBPCRHR2ATMCES1CES2
SCHEMBL7379932 0.76 ATM (0.75) CRHBPCRHR2ATMCES1CES2
SCHEMBL7374227 0.75 CRHBP (0.49) CRHBPCRHR2ATMCES1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed