SCHEMBL7375548

SCHEMBL7375548

COc1ccc(C(=O)CCCCN2CCC(c3ccccc3)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.68
CYP2J2 P51589 1/20 0.66
SIGMAR1 Q99720 2/20 0.64
KMT2A Q03164 2/20 0.59
OPRM1 P35372 1/20 0.57
HTR7 P34969 3/20 0.56
HTR1A P08908 2/20 0.56
HTR2A P28223 2/20 0.56
SLC6A4 P31645 2/20 0.56
HRH1 P35367 2/20 0.56
DRD3 P35462 1/20 0.56
HTR2B P41595 1/20 0.56
MCHR1 Q99705 1/20 0.56
HSD11B1 P28845 1/20 0.56
ALDH1A1 P00352 1/20 0.55
LMNA P02545 1/20 0.55
GAA P10253 1/20 0.55
SLC6A2 P23975 1/20 0.54
HTR2C P28335 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8054055 0.99 DRD2 (0.67) DRD2CYP2J2SIGMAR1KMT2AOPRM1
SCHEMBL11861029 0.83 CYP2J2 (0.94) CYP2J2HRH1
Hydrochloric Acid SCHEMBL11866868 0.82 CYP2J2 (0.92) CYP2J2KMT2AHRH1
SCHEMBL11865078 0.82 CYP2J2 (0.92) CYP2J2HRH1
Hydrochloric Acid SCHEMBL10824127 0.81 DRD2 (0.64) DRD2CYP2J2SIGMAR1KMT2AMCHR1
SCHEMBL20652674 0.81 DRD2 (1.00) DRD2SIGMAR1KMT2AOPRM1HTR1A
Hydrochloric Acid SCHEMBL11867724 0.81 CYP2J2 (0.90) CYP2J2KMT2AHRH1
SCHEMBL7375551 0.81 ALDH1A1 (0.59) DRD2CYP2J2SIGMAR1OPRM1ALDH1A1
Hydrochloric Acid SCHEMBL8054053 0.80 ALDH1A1 (0.58) DRD2CYP2J2SIGMAR1OPRM1HTR7
SCHEMBL14435454 0.79 ALDH1A1 (0.78) DRD2KMT2AHTR7HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995000131-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF CAMBRIDGE NEUROSCIENCE, INCORPORATED (US) 1995-01-05 WO disclosed