SCHEMBL7375552

SCHEMBL7375552

COC(=O)CCC(C#N)(CCC(=O)OC)c1ccc(OC)c(OC)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.64
CASP1 P29466 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.50
CYP3A4 P08684 3/20 0.45
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
ABCB1 P08183 3/20 0.41
CYP3A5 P20815 1/20 0.41
NFE2L2 Q16236 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
ELANE P08246 1/20 0.40
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
TSHR P16473 1/20 0.38
MAPK10 P53779 1/20 0.38
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416817 0.89 HSD17B10 (0.52) HSD17B10CASP1L3MBTL1CYP3A4CYP2C19
SCHEMBL7384417 0.88 HSD17B10 (0.66) HSD17B10CASP1L3MBTL1CYP3A4CYP2C19
SCHEMBL7858782 0.86 CASP1 (0.49) HSD17B10CASP1L3MBTL1CNR2PDE4A
SCHEMBL5498111 0.86 CASP1 (0.49) HSD17B10CASP1PDE4APDE4D
SCHEMBL522321 0.84 CASP1 (0.46) HSD17B10CASP1L3MBTL1CYP3A4CYP2C19
SCHEMBL7415171 0.84 HSD17B10 (0.45) HSD17B10CASP1L3MBTL1CYP3A4CYP2C19
SCHEMBL8607187 0.82 CYP3A4 (0.65) HSD17B10CASP1L3MBTL1CYP3A4CYP2C19
SCHEMBL11818519 0.82 ALDH1A1 (0.47) HSD17B10CASP1L3MBTL1CYP2C19CYP1A2
SCHEMBL3519610 0.81 L3MBTL1 (0.45) HSD17B10CASP1L3MBTL1NFE2L2MAPT
SCHEMBL7744791 0.81 HSD17B10 (0.41) HSD17B10CASP1CYP3A4CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4843081-A Aryl and heteroaryl substituted cycloalkyl compounds RORER PHARMACEUTICAL CORPORATION (US) 1989-06-27 US disclosed
US-4795757-A Bisarylamines RORER PHARMACEUTICAL CORPORATION (US) 1989-01-03 US disclosed
US-3985888-A Methods of inducing sedation using certain spiroalkanone-imides RICHARDSON-MERRELL INC. (US) 1976-10-12 US disclosed
US-3979444-A CENTRAL NERVOUS SYSTEM DEPRESSANTS, HYPOTENSIVES THE UPJOHN COMPANY (US) 1976-09-07 US disclosed