SCHEMBL7375725

SCHEMBL7375725

CCCc1cccc2c(=O)cc(-c3cccc(OCO)c3[N+](=O)[O-])oc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.44
CCNB1 P14635 2/20 0.44
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 4/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 3/20 0.43
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP2D6 P10635 3/20 0.38
LMNA P02545 2/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 3/20 0.34
CYP2C19 P33261 3/20 0.34
TSHR P16473 2/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
NPC1 O15118 1/20 0.34
GMNN O75496 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378571 0.77 ALDH1A1 (0.73) ALDH1A1CYP3A4MAPTHPGDKDM4E
SCHEMBL7375720 0.73 KDM4E (0.46) ALDH1A1CYP3A4HPGDKDM4EHSD17B10
SCHEMBL8405242 0.69 HPGD (0.68) ALDH1A1CYP3A4MAPTHPGDKDM4E
SCHEMBL12835496 0.68 ALDH1A1 (0.58) CDK1CCNB1ALDH1A1CYP3A4MAPT
SCHEMBL12835507 0.67 ALDH1A1 (0.70) ALDH1A1CYP3A4MAPTHPGDKDM4E
SCHEMBL10966059 0.67 MAOB (0.47) MAPTCYP2D6KMT2AHTTGAA
SCHEMBL7379294 0.66 CYP2D6 (0.48) CDK1CCNB1ALDH1A1CYP3A4MAPT
SCHEMBL7373845 0.65 MAPT (0.48) ALDH1A1CYP3A4MAPTHPGDKDM4E
SCHEMBL7087276 0.65 CYP2D6 (0.64) CDK1CCNB1ALDH1A1CYP3A4MAPT
SCHEMBL7374866 0.65 ALDH1A1 (0.53) ALDH1A1CYP3A4MAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115718-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000017184-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2000-03-30 WO disclosed